Relationships between opiate receptor binding and analgetic properties of prodine-type compounds.

نویسندگان

  • W A Klee
  • M A Iorio
چکیده

The receptor binding affinities of some diastereoisomeric prodine analgoues have been compared with their analgetic activities determined by the hot-plate test in mice. The close correlation found between these potencies indicates that the relative analgetic activities of the alpha/beta isomers are determined primarily by the appropriate association to the receptor sites.

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عنوان ژورنال:
  • Journal of medicinal chemistry

دوره 20 2  شماره 

صفحات  -

تاریخ انتشار 1977